Target engagement and drug residence time can be observed in living cells with BRET | Nature Communications
Promega Launches NanoBRET™ Target Engagement Intracellular Kinase Assay, First to Quantitatively Measure Drug-Kinase Interactions in Live Cells | Business Wire
Determining target engagement in living systems | Nature Chemical Biology
Target engagement approaches for pharmacological evaluation in animal models - Chemical Communications (RSC Publishing)
Target engagement approaches for pharmacological evaluation in animal models - Chemical Communications (RSC Publishing) DOI:10.1039/C9CC02824B
CETSA: a target engagement assay with potential to transform drug discovery. | Semantic Scholar
HDAC11 target engagement assay development in cells – CETSA – openlabnotebooks.org
Target Engagement in Lead Generation - ScienceDirect
Determining target engagement in living systems | Nature Chemical Biology
Screening for Target Engagement using the Cellular Thermal Shift Assay - CETSA - Assay Guidance Manual - NCBI Bookshelf
Target Engagement in Lead Generation - ScienceDirect
A Cell-Based Target Engagement Assay for the Identification of Cereblon E3 Ubiquitin Ligase Ligands and Their Application in HDAC6 Degraders - ScienceDirect
Target Engagement in Lead Generation - ScienceDirect
Labelled chemical probes for demonstrating direct target engagement in living systems | Future Medicinal Chemistry
Critical Needs in Cellular Target Engagement | Eurofins DiscoverX Blog
Target Engagement for Drug Discovery
Promega NanoLuc Enables a First in Measuring Drug-Target Residence in Live Cells | Business Wire
Small Molecule Tools to Study Cellular Target Engagement for the Intracellular Allosteric Binding Site of GPCRs - Huber - 2023 - Chemistry – A European Journal - Wiley Online Library